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Metabolism / Catalysis / CYP2A6 / Enzyme kinetics / CYP2D6 / Enzyme / Methoxsalen / Paroxetine / CYP2E1 / Chemistry / Cytochrome P450 / Enzymes


Validation of Mechanism Based Inhibition: Our Experience Franca Pugnaghi, Craig Thomas, Rachael Brown and Peter Fenn Aptuit Limited, Riccarton, Edinburgh EH14 4AP, UK
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Document Date: 2015-02-05 10:57:53


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City

San Diego / Edinburgh / Oxford / Staines / /

Company

Peter Fenn Aptuit Limited / Wilson / Amersham Pharmacia Biotech UK Ltd / Tissue Transformation Technologies / Sigma-Aldrich / In Vitro Technologies / Sequoia Research Products Ltd / Erithacus Software Ltd. / /

Country

United States / United Kingdom / /

Currency

CYP / pence / /

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IndustryTerm

enzyme active site / chemical entities / /

Person

Rachael Brown / Craig Thomas / Chin Pharmacokinet / Franca Pugnaghi / /

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Position

Lopez-Garcia MP / /

Product

M-16 / Experience Methoxsalen - CYP2A6 / /

Technology

Drug Metabolism / /

URL

www.aptuit.com / /

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