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Amines / Organofluorides / Alkynes / Organochlorides / Gefitinib / Erlotinib / Epidermal growth factor receptor / Hsp90 / Protein kinase inhibitor / Chemistry / Organic chemistry / Quinazolines


The HSP90 Inhibitor, AT13387, Displays Single Agent Activity in Erlotinib-Sensitive and -Resistant Models of EGFR-Activated NSCLC Keisha Hearn, Tomoko Smyth, Jon Lewis, Vanessa Martins, Neil Thompson, Mohammad Azab, John
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City

Cambridge / NCI / /

Company

HSP90 / Astex Pharmaceuticals Inc. / Nicola G. Wallis Astex Pharmaceuticals / Wallis Astex Pharmaceuticals / /

Event

FDA Phase / /

MedicalCondition

resistant disease / Cancer / xenograft tumors / tumors / non-small cell lung cancer / NSCLC / EGFR-activated tumor / /

Person

Keisha Hearn / Jon Lewis / Mohammad Azab / Vanessa Martins / Neil Thompson / Tomoko Smyth / John Lyons / /

Product

H1975 / AT13387 / /

Technology

Genotype / /

URL

www.astx.com / /

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