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Imatinib / Piperazines / Pyridines / Pyrimidines / Gastrointestinal stromal tumor / CD117 / Tyrosine kinase / Sunitinib / Hsp90 / Biology / Chemistry / Organic chemistry


The HSP90 inhibitor, AT13387, demonstrates potent anti-tumor activity in both imatinib-sensitive and -resistant gastrointestinal stromal tumor models No A217 Tomoko Smyth1, Thomas Van Looy2, Jayne Curry1, Ana Rodriguez-
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City

Cambridge / /

Company

Astex Pharmaceuticals Inc. / INTRODUCTION 1Astex Pharmaceuticals / /

Country

United Kingdom / Belgium / /

Facility

Women’s Hospital / University Hospitals / Laboratory of Experimental Oncology / Catholic University of Leuven / /

IndustryTerm

Cancer Therapeutics / /

MedicalCondition

tumor / gastrointestinal stromal tumors / necrosis / tumors / resistant gastrointestinal stromal tumor / /

Organization

Women’s Hospital / /

Position

General / /

Technology

Pharmacodynamics / /

SocialTag