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Digoxin / ABC transporters / Torsades de pointes / Antiarrhythmic agent / Amiodarone / IC50 / Dabigatran / P-glycoprotein / Chemistry / Organic chemistry / Cardenolides


The Role of Drug Transporters in Drug Safety-Perspective from the FDA
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City

New Orleans / /

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Event

Product Recall / Product Issues / /

MedicalCondition

Natalizumab* Multiple sclerosis / 99m Tc** Diagnostic aid Cardiopulmonary arrest / Bromfenac NSAID Acute liver failure / Terfenadine Antihistamine Torsades de Pointes / Rapacuronium Anesthesia Bronchospasm / Valdecoxib Pain relief Cholesterol lowering Torsades de Pointes / Troglitazone Diabetes / stroke CYP/transporter substrate Skin reactions / constipation / Astemizole Antihistamine Torsades de Pointes / Chronic / stable angina Torsades de Pointes / Grepafloxacin Antibiotics Risk CYP/transporter inhibitor Torsades de Pointes / Drug-drug interactions Heart attack / Drug-drug interactions Acute liver failure Rhabdomyolysis / women Ischemic colitis / Alosetron* Irritable bowel syndrome / Levomethadyl Opiate dependence Fatal arrhythmia / /

Organization

FDA / office of Planning and Analysis / World Congress / American Association of Pharmaceutical Scientists Annual / office of Clinical Pharmacology / OTS Center for Drug Evaluation and Research / /

Product

clopidogrel / Drugs / simvastatin / digoxin / Technetium / Pemoline / /

Technology

pharmacokinetics / /

URL

http /

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